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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10759 | CEP-28122 mesylate salt (1022958-60-6 free base) | CEP-28122 mesylate salt | ALK |
CEP-28122 mesylate salt (1022958-60-6 free base) is a highly selective orally active ALK inhibitor (IC50: 1.9 nM in an enzyme-based TRF assay). | |||
T72317 | CEP-28122 mesylate salt | ||
CEP-28122 mesylate salt, a diaminopyrimidine derivative, serves as a potent, selective, and orally bioavailable ALK (anaplastic lymphoma kinase) inhibitor, exhibiting an IC 50 value of 1.9 nM against recombinant ALK kina... |